Opioids, Part 1Huda Akil, Albert Herz, Eric J. Simon |
Contents
CHAPTER | 3 |
E Putative Endogenous Ligands | 9 |
G Recent Studies on Purified μOpioid Binding Protein | 18 |
Copyright | |
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8-binding Acad Sci USA adenylate adenylyl cyclase adrenal affinity agonist amino acid analgesic analogs antinociception binding sites Biochem Biol Chem bovine brain membranes Brain Res cells CH₂O cortex cyclic d-receptors deferens dopamine DPDPE drugs dynorphin effects enkephalin enzyme function G protein gene expression glucocorticoids guanine guanine nucleotides guinea pig Herz Höllt hypothalamus immunoreactivity increase inhibition inhibitors interaction K-sites kappa Kosterlitz HW ligands lobe mediated modulation Mol Pharmacol morphine mouse mRNA mRNA levels naloxone naltrexone Natl Acad Sci Neurochem neurons Neuropeptides Neurosci neurotransmitter nucleotides nucleus nucleus accumbens opiate receptors opioid agonists opioid binding opioid peptides PDYN PENK gene PENK mRNA Pharmacol Exp Ther pharmacological pituitary POMC POMC gene POMC mRNA Portoghese potent precursor presynaptic Proc Natl Acad ProDyn proenkephalin proopiomelanocortin rat brain receptor complex regulation release ROTHMAN selective sequence slices specific spinal cord ẞ-endorphin stimulation striatal striatum structure studies synthesis tissue transcription treatment vas deferens vitro vivo