Peptidergic G Protein-coupled Receptors: From Basic Research to Clinical ApplicationsPierangelo Geppetti, Werner Müller-Esterl, Domenico Regoli |
Contents
Preface | 1 |
Posttranslational Modifications of Endothelin Receptors Modulate Signal Transduction | 29 |
Discovery and Design of Peptide and NonPeptide Ligands to G ProteinCoupled | 52 |
Copyright | |
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affinity agonist airways antibodies arrestin asthma autoradiography B₁ B₂ binding sites Biol biological bradykinin receptor bronchoconstriction capsaicin CCKA antagonists CCKA receptor Chem chemokine clinical cloned compounds coupled CXCR4 desensitization devazepide disease domain DRGs effect endogenous endothelin enteric neurons ETA and ETB ETB receptor excitatory expression functional G protein-coupled receptors G-protein gallbladder gastric emptying gastrin Gastroenterology gastrointestinal gene Geppetti GPCR GRK2 human increase induced inflammation inflammatory inhibition inhibitory interaction intracellular kinin kinin receptors ligand loxiglumide mechanisms mediated membrane molecular mRNA mutant myenteric N-terminus nerve neurokinin neuropeptide Neuroscience nitric oxide nociceptin non-peptide palmitoylation pancreatic pathway patients peptide Pharmacol pharmacological phosphorylation Physiol plasma extravasation potential proteases protein-coupled receptors pulmonary Rat Brain receptor activation receptor antagonist receptor autoradiography receptor binding receptor kinase receptor subtypes Regoli regulation release residues response role Rovati secretion smooth muscle specific stimulation studies tachykinins thrombin tissues vitro vivo