Sulphur Containing Drugs and Related Organic Compounds: Metabolism and pharmacokinetics of sulphur containing drugs, pt. A-B. (2v.)L. A. Damani |
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6-mercaptopurine 6-thioguanine 6TGN concentrations absorption acid activity agents allopurinol Andreasen angiotensin-converting enzyme antithyroid drugs assay azathioprine bioavailability Biochem biological fluids blood captopril carbimazole Chem chemical Chromatogr chronic clearance Clin clinical compounds conjugates cysteine cytotoxic dapsone desulphuration detection disulfiram effect elimination half-life Elion ethionamide ethionamide and prothionamide formation glutathione hepatic high performance liquid HPLC human Hyperthyroid inhibition inhibitor intravenous Lennard leukaemia liquid chromatography liver malathion Marchant metabolism and pharmacokinetics metabolites methimazole methods mg/kg mixed disulphide nucleotide oral administration oral dose oxidation patients penicillamine penicillamine disulphide Pharm pharmacokinetics Pharmacol pharmacology plasma concentrations plasma proteins propylthiouracil protein binding prothionamide purine pyrithione radioactivity reactions red cell renal reported riboside S-methyl sensitive serum Skellern skin spironolactone studies sulphate sulphoxide sulphur sulphur-containing Taurog Ther therapeutic thioamides thiobarbiturates thiocarbamide thioinosinic thiol thiopental thiopentone thiopurine drug thyroid tissue toxicity Toxicol uptake urine vitro vivo volume of distribution