Current Medicinal Chemistry |
Common terms and phrases
acetylation activity adducts Agents Guest Editor analogues antagonist anti antibodies antiestrogens arylamines assays autophosphorylation Bentham Science Publishers binding bioactivation biological breast cancer breast tumour calmodulin CaM antagonism CaM dependent carcinogenic cascade catalyze cellular clinical compounds conformation covalent cytotoxicity dapsone detoxification dimerization drug effect effector EGFr EGFr family enzyme estrogen formation function genes glycosylated growth factor heterocyclic amines heterodimerization heterodimers hormone human hydroxylamine idoxifene immune increased induced inhibition inhibitors interactions juxtamembrane knockout lCso leukocytes ligands macrophages MAP kinase mechanism Medicinal Chemistry membrane metabolic metabolites mice microsomal mitogenesis mitogenic monocytes murine mutations NAT1 NAT2 oncogenes overexpressing pathway patients peptide phenotype phosphorylation PMNs potency procainamide proliferation protein reaction receptor residues retro-inverso RTKs SH2 domain signaling slow acetylators structure substrate suggest sulfamethoxazole sulfonamide synthesis Tamoxifen TGF-a therapeutic tissues toxicity transformed tuftsin tuftsin analogs tumour type l RTKs tyrosine kinase vitro vivo